平安! 发表于 2011-11-9 19:57 0 p5 [- }3 a. U9 o
Pazopanib (100 mg/kg/day free base equivalent) & B5 W" @; x* Z* D- |+ u$ A
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
; h2 b8 G7 K! {5 h% S# E+ {搜索了一下,原料一大堆。
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, p. }, @0 U# `3 ]对不起!100mg/kg是用于移植瘤的,我弄错了。3 ~( v, l2 K: z6 Q7 b# l" N ^
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以下是正版说明书的推荐用量。9 ~- O9 I6 P p, H& q, B. a
8 E6 J+ i6 N( t& V, R9 C--------------------- DOSAGE AND ADMINISTRATION ----------------
. ?8 ]# ]! S; g4 P+ e: I7 H) u* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) 4 O" [) d5 r: m: J" ^+ t- o" m
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 1 ?$ T4 c! N8 q6 P `' v$ n1 S7 N
---------------------DOSAGE FORMS AND STRENGTHS --------------- _9 Q8 n I- J' J- w1 J! N
200 mg tablets. (3) , ~' }& O/ s" m8 l8 L+ z( g
-------------------------------CONTRAINDICATIONS------------------------ |